共查询到19条相似文献,搜索用时 93 毫秒
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刘立伟 《河北北方学院学报(自然科学版)》2019,35(10)
水飞蓟素具有多种药理活性,除保肝护肝作用外,对肿瘤、糖尿病、阿尔茨海默症等神经系统疾病也有较好治疗效果,是一种重要的医药原料。水飞蓟素多采用常温浸渍、碱提酸沉、超声和回流等方法提取,近年来涌现出超临界流体提取法、酶法、双水相萃取法、亚临界低温萃取法等新型提取方法。综述了水飞蓟素的提取方法及药理活性,以期为更好开发和利用水飞蓟资源提供参考。 相似文献
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【目的】观察接种致死量鸭肝炎病毒后雏鸭生长及发育的改变及水飞蓟素对其的影响。【方法】100只11日龄雏鸭分为5组,分别为攻毒组、攻毒+30 mg水飞蓟素组、攻毒+10 mg水飞蓟素组、10 mg水飞蓟素组、空白对照组。试验期内正常喂食及饮水,并每隔3 d空腹测定一次体重,观察动物发病及死亡情况。于攻毒后的第15 d和第30 d测定动物吻尾长度,于攻毒后第30 d扑杀,并测定腹脂重以及各内脏器官指数。【结果】用致死量鸭肝炎病毒攻击后,雏鸭在96 h内死亡严重,死亡率达75%(第1组);30、10 mg?kg-1bw?d-1的水飞蓟素具有良好的保护作用,死亡率分别为20%和0(第2组,第3组)。第1、第2组的幸存者显示出显著快的增重和发育速度,胴体构成发生了明显改变,内脏指数显著降低,胸肌指数显著上升。10 mg?kg-1bw?d-1的水飞蓟素可有效抑制病毒的促生长发育效应,但30 mg?kg-1bw?d-1的水飞蓟素却没有抑制效应。【结论】致死量鸭肝炎病毒可显著促进存活雏鸭的生长发育,水飞蓟素对鸭肝炎病毒的促生长发育效应具有双相性作用,在较低剂量时可发挥抑制作用,但在较高剂量时抑制作用丧失。 相似文献
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以菊科植物水飞蓟为试验材料,采用浓度为50、100、200、300、400 mmol/L的NaCl溶液分别对水飞蓟进行盐处理,研究不同盐浓度对水飞蓟素含量的影响.结果表明,NaCl溶液浓度在50~400mmol/L范围内水飞蓟素含量随着盐浓度的升高有所增加. 相似文献
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对水飞蓟资源、化学成分、提取工艺及水飞蓟油药理活性等方面的研究进展进行了综述,并提出了开发利用水飞蓟油的建议。 相似文献
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对水飞蓟组织培养中外植体来源、愈伤组织诱导、再生植株诱导、毛状根诱导以及组织培养物中活性成分等方面进行了综述,以期为解决水飞蓟的资源需求以及以组织培养为基础的基因与代谢工程研究提供理论及技术指导。 相似文献
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高寒地区水飞蓟高产栽培技术 总被引:1,自引:0,他引:1
闫振宏 《农村实用科技信息》2012,(4):30
水飞蓟是一种菊科药用作物,是北药中的一个品种,喜温暖阳光充足环境,耐寒、耐贫瘠土地,是作物调茬的好品种。水飞蓟种子内含水飞蓟素,水飞蓟素是制作保肝利胆药品的主要原料,它的主要功能是清热解毒、保肝、利胆、保脑,可使肝脏患者自觉症状和某些生化指数如血清胆红素、白朊及球朊系数、凝血酶元、谷丙转氨酶等迅速改善。同时种子含油量一般为28~36%,食用此油又可防止动脉硬化。由于近几年水飞蓟市场行情好,当季效益高,而且 相似文献
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水飞蓟,别名水飞雉、奶蓟、老鼠筋、乳蓟子等,为菊科1-2年生草本植物,1972年从德国引入我国。其成熟的种子具有很高的药用、食用及经济价值,用途非常广泛,具有清热解毒、保肝护肝、利胆、健脑和抗辐射的功能,从该植物种子中提取的水飞蓟素是制造西里马灵、益肝灵、水飞蓟素片、利肝片、保肝宁、飞当片等中成药的重要原料. 相似文献
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LIU Wei-min WANG Bing-yun CHEN Jian-hong WANG Jun JI Hui-qin YUAN Sheng HUANG De-chun LI Kang-lin 《中国农业科学(英文版)》2009,8(11):1403-1408
To evaluate the effects of duck hepatitis virus-1 (DHV-1) on the body weight gain in duck and the effects of silymarin on it in vivo, 100 10-d-old ducks, both male and female, were collected to be subjected to the test. The experiments were conducted in 8 groups: in group 1-3, the animals were inoculated with 1:105 diluted duck hepatitis virus (DHV-1) infected allantoic fluid and given 0, 30, and 50 mg kg^-1 BW d^-1 silymarin orally, respectively. In group 4-6, the animals were inoculated with 1:5 × 105 diluted DHV-1 infected allantoic fluid and given 0, 10, and 30 mg kg^-1 BW d^-1 silymarin orally, respectively. In group 7, the animals were given 10 mg kg^-1 BW d^-1 silymafin only. Group 8 was the control one treated by injecting sterillized saline into the leg muscles. All the silymarin was given from 0 to 4 d after inoculation of the virus. By the 5th d after inoculation, the vein blood was drawn from the dorsal foot vein and the plasma samples were collected and stored at -20℃. The body weight gain (BWG) was measured from 0 to 10 d after inoculation. The plasma IGF-I, T3, and T4 concentrations were measured by radioimmunoassay (RIA). At the virus dose of 1:5 ×105 diluted virus infected allantoic fluid, the inoculation of the virus enhanced the BWG significantly compared with that of the control (P〈 0.01), while 10-50 mg kg^-1 BW d^-1 silymarin could counteract the effects of the virus on the BWG dose-dependently. The plasma IGF-I levels showed no correlation with the BWG, but the T3 levels showed a same tropism with the body weight gain. The present results indicated that sublethal DHV-1 enhanced the body weight gain of ducklings significantly, and the silymarin could counteract this effect in vivo. 相似文献
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S. V. Lutsenko T. V. Kashnikova A. V. Khmyrov E. A. Druz’ O. N. Ledeshkova N. B. Fel’dman N. D. Luzhnov E. V. Lutsenko 《Russian Agricultural Sciences》2008,34(6):415-417
A liposomal form of silymarin has been produced. The preparation promotes growth of muscle tissue and has a positive effect on the chemical composition and quality of meat, increasing the dry matter, fat, and total protein content in breast meat. 相似文献
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The kinetic mechanism for the preparation of silymarin from milk thistle seeds was studied during the microwave-assisted extraction (MAE) process. The results showed that the transfer rate of silymarin from milk thistle seeds increased with the microwave output power and temperature during MAE processing. The apparent extraction rate constant k (s?1) was 1.2028×10?2, 1.2248×10?2, and 1.2485×10?2, and diffusion coefficient D (m2 ? s?1) was 4.21×10?10, 4.29×10?10, and 4.37×10?10 at the microwave temperatures of 383, 393, and 403 K, respectively, in the silymarin MAE process. With the help of scanning electron microscopy (SEM), the microstructures of the samples extracted by MAE were observed. The results revealed that the increased efficiency and rate of MAE of silymarin could be attributed mainly to the subsequent cell change resulting from superheating effects during MAE. 相似文献
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[目的]考察不同水飞蓟种子处理方法对植株生长及所结果实中水飞蓟素含量的影响,确定种子的最佳处理方法。[方法]将水飞蓟种子分别经冷藏、冷冻等方法处理后播种,考察种子的发芽率、株高、株幅、现蕾时间及单株产量,并比较所结果实中水飞蓟素的含量,筛选种子的最佳处理方法。[结果]水飞蓟种子经超低温处理后播种发芽率最低,生长最弱,果实中水飞蓟素含量最低;自然越冬处理(秋季播种)的种子萌发后长势好,产量最高,且所结果实中水飞蓟素的含量最高。[结论]水飞蓟种子在秋季播种后植株的生长状况较好,产量高,值得进一步研究和推广。 相似文献
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目的了解辛伐他丁对2型糖尿病大鼠血管内皮细胞黏附分子-1(VCAM-1)和单核细胞趋化因子-1(MCP-1)的影响。方法30只SD大鼠随机分为正常组(NC)、糖尿病组(DMC)、辛伐他丁治疗组(DMT),每组各10只大鼠。喂养12周后抽血测定血脂全套,取主动脉标本以免疫组化和半定量RT-PCR法分别检测VCAM-1和MCP-1的mRNA和蛋白表达。结果DMT组大鼠血管内皮VCAM-1和MCP-1的mRNA和蛋白表达明显降低,与DMC组比较差异有统计学意义(P<0.05)。结论辛伐他丁可减少糖尿病大鼠血管内皮VCAM-1和MCP-1的表达,减轻血管内皮局部的炎症反应。 相似文献
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目的 观察罗格列酮对2型糖尿病大鼠骨骼肌解偶联蛋白3(UCP3)、肉碱棕榈酰转移酶-I(CPT—I)mRNA表达及疗效的影响。方法58只SD大鼠随机分为普通饲养组(NC组,n=15)、高脂饲养组(HF组,n=15)和糖尿病组。糖尿病组大鼠在高脂饲料喂养至8周末时,腹腔注射链唑霉素(25mg/kg)制作糖尿病模型;再随机分为糖尿病治疗组(DMT组,n=14)和糖尿病未治疗组(DMC组n=14),分别给予罗格列酮(3mg·kg^-1·d^-1)和灭菌生理盐水灌胃,持续8周。UCP3、CPT—ImRNA表达采用RT—PCR测定。结果HF与DMC组骨骼肌UCP3、CFT—ImRNA表达明显低于NC组(P〈0.05)。与DMC组比较,DMT组血糖和游离脂肪酸降低,而胰岛素敏感性和骨骼肌UCP3、CFT-ImRNA表达增加(P〈0.05)。结论2型糖尿病大鼠骨骼肌UCP3、CPT—InLRNA表达降低;而罗格列酮可上调UCP3、CFT—ImRNA的表达,降低血糖、FFA水平。 相似文献
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观察糖康抗氧化应激对实验性糖尿病大鼠视网膜病变的疗效并探讨其作用机制。采用腹腔注射链脲佐菌素(STZ)复制糖尿病模型并随机分为正常对照组、模型组、糖康高、中和低剂量组和达纳康组,每日灌胃,定期检测大鼠体重和非空腹血糖;第12周末,消化铺片法观察视网膜微血管病理和形态学改变;化学比色法检测各组大鼠血清及视网膜组织中超氧化物歧化酶(SOD)活性和丙二醛(MDA)含量。与正常组比较,模型组血清及视网膜SOD活性明显降低(P0.01),MDA含量明显升高(P0.01),无细胞毛细血管条索数明显升高,约为正常组的5.33倍(P0.01);与模型组比较,各治疗组均可提高血清及视网膜SOD活性,降低MDA含量,且以糖康高剂量组最为显著(P0.01),无细胞毛细血管条索数明显降低(P0.01)。糖康可显著降低糖尿病大鼠的氧化应激水平,提高糖尿病大鼠血清及视网膜的抗氧化能力。 相似文献