New Algorithms for Data Discretization Based on Rough Set Theory

The discretization of real values is always one of the key problems to be solved in the domain of machine learning for its great contribution to speeding up the followed learning algorithms, cutting down the real demand of algorithms on running space and time, and improving the clustering capability of the ultimate learning results. The basic characteristics and framework of discretization approaches based on rough set model are analyzed at first, then the different measurements of the importance of candidate cuts are discussed and researched. Two new heuristic algorithms are put forward to finally select the useful cuts from a candidate set. The selected cuts of the two algorithms will adequately maintain the discernible relation of information systems for their full considering the specialty of rough set, which perfectly embodies the advantages of this theory. Moreover, excellent discretization results may be expected through these heuristic algorithms.     

COUPLING ANALYSIS METHOD FOR INTERACTION BETWEEN FOUNDATION WITH CAVERN AND FRAME STRUCTURE

In this paper,the interaction between foundation withcavern and frame structure is studied by the coupling methods of BEMand FEM.On the interface between the foundation and structure,thecoupling analysis needs to satisfy both the condition of displacementcompatibility and force equilibrum.A calculating program for two-dim-ensional problem is worked out in the computer,SIEMENS 7570C.Twoengineering examples are calculated and the results are compared withthose obtained by the comventional simplified method and with the observedresults from the engieering structures.It indicates that it is necessaryfor the weak rock foundation with shallow cavern,in the buried depth,to take the interaction into account.     

面粉品质性状与速冻水饺品质关系的研究

对7种面粉的化学成分、面团流变学特性等指标进行测定,详细分析了各项指标与速冻水饺品质的相关关系,得出适合生产速冻水饺的面粉的最佳特性指标。并通过比较分析对黑龙江省地产小麦粉生产速冻水饺的适用性进行评价。     

Structural Effects of N-Arylcarbamoylpyrazolines on Calcium Uptake in Rat Brain Synaptosomes

N-Arylcarbamoylpyrazolines with various substituents at the para position of the carbamoyl benzene ring inhibited ATP-dependent Ca²⁺-uptake in synaptosomes prepared from the rat brain. The activity of these compounds was evaluated as log(1/I₅₀), the reciprocal logarithm of half inhibitory concentration, I₅₀ (m ), from the concentration–response curve for the inhibition of Ca²⁺-uptake. Among the compounds tested, methyl 3-(4-chlorophenyl)-4-methyl-1-[N-(4-trifluoromethylphenyl)carbamoyl]-2-pyrazoline-4-carboxylate was the most potent, the I₅₀ value of which as 9·12×10⁻⁷ m . Variations in the activity in terms of log(1/I₅₀) were quantitatively analysed using a substituent parameter, showing that the higher the electron-withdrawing effect of the substituent, the higher was the activity. The substituent effects were similar to those on insecticidal activity against the Americal cockroach. The higher the inhibitory activity against Ca²⁺ uptake, the higher seemed to be the insecticidal activity. Methyl(4S) - 3 - (4 - chlorophenyl) - 4 - methyl - 1 - [N - (4 - chlorophenyl)carbamoyl] - 2 - pyrazoline -4-carboxylate had higher inhibitory activity against Ca²⁺-uptake and higher in-secticidal activity than the R-isomer, but the difference was greater in theCa²⁺-uptake system.     

Synthesis and Structure–Activity Relationships of Miticidal 4,5-Dihydropyrazole-5-thiones

A series of novel 4,5-dihydropyrazole-5-thiones (DHPs) was synthesised by treating the corresponding dihydropyrazolones with ‘Lawesson’s reagent and evaluated for miticidal activity against two-spotted spider mites (Tetranychus urticae Koch). Of these, 3-(4-chlorophenyl)-4,4-dimethyl-1-phenyl-4,5-dihydropyrazole-5-thione, 3-(4-chlorophenyl)-4-ethyl-4-methyl-1-phenyl-4,5-dihydropyrazole-5-thione, 3-(4-chlorophenyl)-1-phenyl-4,5-dihydropyrazole-5-thione-4-spirocyclopentane and 4,4-dimethyl-1-phenyl-3-(4-trifluoromethyl-phenyl)-4,5-dihydropyrazole-5-thione were highly active (pEC₅₀>4·0) and were more effective than the miticide dicofol (pEC₅₀=3·879), which has traditionally been used for the control of phytophagous mites. Structure–activity relationship (SAR) studies were performed on each position of the pyrazole ring of DHPs. The results indicated that the unsubstituted phenyl, 4-substituted phenyl and thioxo groups on the 1-, 3- and 5-positions of DHPs respectively were required for activity. Quantitative SAR studies using physicochemical parameters of substituents and the capacity factor k′ as a hydrophobicity index suggested that: (a) the activities of all types of DHPs examined were mainly dominated by hydrophobicity, (b) the bulkiness of 4-substituents of the 3-phenyl ring favoured the activity and (c) the log k′ optimum for all DHPs was 1·675, equivalent to a log P_ow value of c. 5·0.     

荔枝空中压条苗根系生长动态及与地上部生长的相互关系

以‘糯米糍’荔枝Litchi chinensis Sonn．空中压条苗为试材,利用根箱栽培研究了周年内3株荔枝幼树根系形态、动态生长以及与地上部枝梢生长间的相互关系．结果表明：荔枝不同类型的根在形态上差异较大,侧根粗壮发达,生长周期长,可持续生长8～10周;须根纤细茂密,寿命只有2～3周．2株苗的根系周年内有2次大的生长峰和2次小的生长峰,根梢生长表现为交替生长．1株苗在周年内只有1次大的生长峰和4次小的生长峰,根梢生长表现为同步生长．3株幼树根梢比值均在1．0左右,表明地上和地下部等量生长．根系生长峰的出现主要表现为新根数量的增加而非原有根系的延长生长．